Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase pim-1' and Ligand = 'BDBM108339'   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Serine/threonine-protein kinase pim-1 (Homo sapiens (Human))	BDBM108339 (US8604217, 343) Show SMILES CN(C)CCN1CCN(CC1)c1nc2c(Br)c(Br)c(Br)c(Br)c2[nH]1 Show InChI InChI=1S/C15H19Br4N5/c1-22(2)3-4-23-5-7-24(8-6-23)15-20-13-11(18)9(16)10(17)12(19)14(13)21-15/h3-8H2,1-2H3,(H,20,21)	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	36.8	n/a	n/a	n/a	n/a	7.0	n/a
Selvita S.A. US Patent					Assay Description Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...				US Patent US8604217 (2013) BindingDB Entry DOI: 10.7270/Q2RJ4H31
					More data for this Ligand-Target Pair