Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase pim-1' and Ligand = 'BDBM108363'   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Serine/threonine-protein kinase pim-1 (Homo sapiens (Human))	BDBM108363 (US8604217, 58) Show SMILES Brc1c(Br)c(Br)c2[nH]c(NCCCN3CCCC3)nc2c1Br Show InChI InChI=1S/C14H16Br4N4/c15-8-9(16)11(18)13-12(10(8)17)20-14(21-13)19-4-3-7-22-5-1-2-6-22/h1-7H2,(H2,19,20,21)	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	25.7	n/a	n/a	n/a	n/a	7.0	n/a
Selvita S.A. US Patent					Assay Description Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...				US Patent US8604217 (2013) BindingDB Entry DOI: 10.7270/Q2RJ4H31
					More data for this Ligand-Target Pair