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Found 1 hit Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase pim-1' and Ligand = 'BDBM108373'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Serine/threonine-protein kinase pim-1


(Homo sapiens (Human))
BDBM108373
PNG
(US8604217, 90)
Show SMILES NCC(O)CNc1nc2c(Br)c(Br)c(Br)c(Br)c2[nH]1
Show InChI InChI=1S/C10H10Br4N4O/c11-4-5(12)7(14)9-8(6(4)13)17-10(18-9)16-2-3(19)1-15/h3,19H,1-2,15H2,(H2,16,17,18)
PDB
MMDB

KEGG

UniProtKB/SwissProt

B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem

Similars

US Patent
n/an/a 13.1n/an/an/an/a7.0n/a



Selvita S.A.

US Patent


Assay Description
Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...


US Patent US8604217 (2013)


BindingDB Entry DOI: 10.7270/Q2RJ4H31
More data for this
Ligand-Target Pair