Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase pim-1' and Ligand = 'BDBM108413'   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Serine/threonine-protein kinase pim-1 (Homo sapiens (Human))	BDBM108413 (US8604217, 372) Show SMILES CNCCCN(Cc1ccccc1)c1nc2c(Br)c(Br)c(Br)c(Br)c2[nH]1 Show InChI InChI=1S/C18H18Br4N4/c1-23-8-5-9-26(10-11-6-3-2-4-7-11)18-24-16-14(21)12(19)13(20)15(22)17(16)25-18/h2-4,6-7,23H,5,8-10H2,1H3,(H,24,25)	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	45.2	n/a	n/a	n/a	n/a	7.0	n/a
Selvita S.A. US Patent					Assay Description Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...				US Patent US8604217 (2013) BindingDB Entry DOI: 10.7270/Q2RJ4H31
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