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Found 1 hit Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase pim-1' and Ligand = 'BDBM50260544'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Serine/threonine-protein kinase pim-1


(Homo sapiens (Human))		BDBM50260544
PNG
(CHEMBL4062679)
Show SMILES NC1CCN(CC1)c1ccc(cc1)-c1ccc2c(c[nH]c2c1)-c1ccc(N)nc1F
Show InChI InChI=1S/C24H24FN5/c25-24-20(7-8-23(27)29-24)21-14-28-22-13-16(3-6-19(21)22)15-1-4-18(5-2-15)30-11-9-17(26)10-12-30/h1-8,13-14,17,28H,9-12,26H2,(H2,27,29)
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MMDB

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Similars
Article
PubMed
n/an/a 2n/an/an/an/an/an/a



Zarqa University

Curated by ChEMBL


Assay Description
Inhibition of human recombinant PIM1 in presence of ATP by ELISA based spectrophotometric analysis

Bioorg Med Chem 25: 4855-4875 (2017)


Article DOI: 10.1016/j.bmc.2017.07.036
BindingDB Entry DOI: 10.7270/Q2BC420V
More data for this
Ligand-Target Pair