Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Serine protease 1/Trypsin-2 (Homo sapiens (Human)) | BDBM50087910 (4-Bromo-N-diaminomethylene-benzenesulfonamide | CH...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem | PubMed | 1.23E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi Curated by ChEMBL | Assay Description Inhibitory activity against human trypsin (using Chromozym TH as the substrate) | J Med Chem 43: 1793-806 (2000) BindingDB Entry DOI: 10.7270/Q2NZ88B0 | |||||||||||
More data for this Ligand-Target Pair |