Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Short transient receptor potential channel 4 (Homo sapiens) | BDBM50529421 (CHEMBL4530872) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | 290 | n/a | n/a | n/a | n/a | n/a | n/a |
Goldfinch Bio Inc. Curated by ChEMBL | Assay Description Inhibition of Englerin-activated human TRPC4 channel expressed in HEK293 cells by Q-patch clamp assay | ACS Med Chem Lett 10: 1579-1585 (2019) Article DOI: 10.1021/acsmedchemlett.9b00430 BindingDB Entry DOI: 10.7270/Q2DN48HF | |||||||||||
More data for this Ligand-Target Pair |