Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sigma non-opioid intracellular receptor 1 (Homo sapiens (Human)) | BDBM50029788 (8-[1-(3,4-Dichloro-phenyl)-meth-(E)-ylidene]-5-(3-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 65.3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Diabetes and Digestive and Kidney Diseases Curated by ChEMBL | Assay Description Ability to inhibit [3H]-(+)-pentazocine binding to guinea pig brain Sigma receptor type 1 | J Med Chem 38: 4776-85 (1996) BindingDB Entry DOI: 10.7270/Q2XW4HVW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma non-opioid intracellular receptor 1 (Homo sapiens (Human)) | BDBM50029788 (8-[1-(3,4-Dichloro-phenyl)-meth-(E)-ylidene]-5-(3-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 65.3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Diabetes and Digestive and Kidney Diseases Curated by ChEMBL | Assay Description Inhibition of [3H]-(+)-pentazocine binding to sigma receptor of guinea pig brain | J Med Chem 37: 3163-70 (1994) BindingDB Entry DOI: 10.7270/Q2F18XSH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma non-opioid intracellular receptor 1 (Homo sapiens (Human)) | BDBM50029788 (8-[1-(3,4-Dichloro-phenyl)-meth-(E)-ylidene]-5-(3-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 65.3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Diabetes and Digestive and Kidney Diseases Curated by ChEMBL | Assay Description Ability to inhibit [3H]-(+)-pentazocine binding to guinea pig brain Sigma receptor type 1 | J Med Chem 38: 4776-85 (1996) BindingDB Entry DOI: 10.7270/Q2XW4HVW | |||||||||||
More data for this Ligand-Target Pair |