Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Signal transducer and activator of transcription 5A' and Ligand = 'BDBM50267876'   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Signal transducer and activator of transcription 5A (Homo sapiens (Human))	BDBM50267876 (CHEMBL4080740) Show SMILES OP(O)(=O)Oc1ccc(CNC(=O)COc2ccc(cc2)C(=O)Nc2ccc(Br)cc2)cc1OP(O)(O)=O Show InChI InChI=1S/C22H21BrN2O11P2/c23-16-4-6-17(7-5-16)25-22(27)15-2-8-18(9-3-15)34-13-21(26)24-12-14-1-10-19(35-37(28,29)30)20(11-14)36-38(31,32)33/h1-11H,12-13H2,(H,24,26)(H,25,27)(H2,28,29,30)(H2,31,32,33)	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	8.60E+3	n/a	n/a	n/a	n/a	n/a	n/a
Institute of Organic Chemistry, Leipzig University, Johannisallee 29, 04103 Leipzig, Germany. Curated by ChEMBL					Assay Description Displacement of 5-carboxyfluorescein-GY(PO3H2)LVLDKW from STAT5A SH2 domain (unknown origin) pretreated for 1 hr followed by fluorescent tracer addit...				Bioorg Med Chem 25: 3871-3882 (2017) Article DOI: 10.1016/j.bmc.2017.05.039 BindingDB Entry DOI: 10.7270/Q26Q20RB
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