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Found 1 hit Enz. Inhib. hit(s) with Target = 'Small conductance calcium-activated potassium channel protein 1/2/3' and Ligand = 'BDBM50092131'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Small conductance calcium-activated potassium channel protein 1/2/3


(Rattus norvegicus-RAT-Rattus norvegicus (Rat))		BDBM50092131
PNG
(1,7-diazonia-15,21-diazapentacyclo[20.6.2.27,14.08...)
Show SMILES C1CCN[c+]2ccn(CCCCCn3cc[c+](NCC1)c1ccccc31)c1ccccc21
Show InChI InChI=1S/C28H34N4/c1-7-17-29-25-15-21-31(27-13-5-3-11-23(25)27)19-9-2-10-20-32-22-16-26(30-18-8-1)24-12-4-6-14-28(24)32/h3-6,11-16,21-22,29-30H,1-2,7-10,17-20H2/q+2
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Article
PubMed
n/an/a 2n/an/an/an/an/an/a



Aristotelian University of Thessaloniki

Curated by ChEMBL


Assay Description
Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activity

Bioorg Med Chem Lett 14: 4231-5 (2004)


Article DOI: 10.1016/j.bmcl.2004.06.011
BindingDB Entry DOI: 10.7270/Q2FF3W4T
More data for this
Ligand-Target Pair