Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Small conductance calcium-activated potassium channel protein 3 (Homo sapiens (Human)) | BDBM50264072 (2-(2-(pyridin-2-ylmethyl)thiazol-4-yl)pyridine | C...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Bristol Myers Squibb Co. Curated by ChEMBL | Assay Description Inhibition of Kca2.3 channel expressed in HEK293 cells by thallium flux assay | Bioorg Med Chem Lett 18: 5316-9 (2008) Article DOI: 10.1016/j.bmcl.2008.08.023 BindingDB Entry DOI: 10.7270/Q2N87BP1 | |||||||||||
More data for this Ligand-Target Pair |