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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Sodium channel protein type 2 subunit alpha' and Ligand = 'BDBM50043996'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Sodium channel protein type 2 subunit alpha


(Rattus norvegicus)		BDBM50043996
PNG
(9H-Fluorene-9-carboxylic acid [3-(2,6-dimethyl-pip...)
Show SMILES CC1CCCC(C)N1CCCNC(=O)C1c2ccccc2-c2ccccc12
Show InChI InChI=1S/C24H30N2O/c1-17-9-7-10-18(2)26(17)16-8-15-25-24(27)23-21-13-5-3-11-19(21)20-12-4-6-14-22(20)23/h3-6,11-14,17-18,23H,7-10,15-16H2,1-2H3,(H,25,27)
PDB
MMDB

KEGG

UniProtKB/SwissProt

B.MOAD
GoogleScholar
AffyNet 
CHEMBL
PC cid
PC sid
UniChem
PubMed
n/an/a 2.90E+4n/an/an/an/an/an/a



Warner-Lambert Company

Curated by ChEMBL


Assay Description
Inhibition of veratridine-induced Na+ influx in chinese hamster ovary cells expressing alpha subunit of rat brain type voltage-gated sodium channel t...

J Med Chem 37: 268-74 (1994)


BindingDB Entry DOI: 10.7270/Q2CJ8F39
More data for this
Ligand-Target Pair