Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sodium channel protein type 8 subunit alpha (Rattus norvegicus) | BDBM50133778 (2,4(5)-Diphenylimidazole | 2,4-diphenyl-1H-imidazo...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 3.22E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Parma Curated by ChEMBL | Assay Description Inhibition of rat NaV1.6-mediated current expressed in human HEK293 cells by patch clamp assay | Bioorg Med Chem Lett 22: 6401-4 (2012) Article DOI: 10.1016/j.bmcl.2012.08.067 BindingDB Entry DOI: 10.7270/Q2TX3GGK | |||||||||||
More data for this Ligand-Target Pair |