Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Sodium channel protein type 9 subunit alpha' and Ligand = 'BDBM254124'   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Sodium channel protein type 9 subunit alpha (Homo sapiens (Human))	BDBM254124 (US9481677, 79) Show SMILES Fc1cc(ccc1Oc1ccc(Cl)cc1-c1ccc2oc(=O)[nH]c2c1)S(=O)(=O)Nc1ncccn1 Show InChI InChI=1S/C23H14ClFN4O5S/c24-14-3-6-19(16(11-14)13-2-5-21-18(10-13)28-23(30)34-21)33-20-7-4-15(12-17(20)25)35(31,32)29-22-26-8-1-9-27-22/h1-12H,(H,28,30)(H,26,27,29)	PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	10.8	n/a	n/a	n/a	n/a	n/a	n/a
XENON PHARMACEUTICALS INC. US Patent					Assay Description Patch voltage clamp electrophysiology allows for the direct measurement and quantification of block of voltage-gated sodium channels (Nav's), and...				US Patent US9481677 (2016) BindingDB Entry DOI: 10.7270/Q20V8BQT
					More data for this Ligand-Target Pair