Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sodium channel protein type 9 subunit alpha (Homo sapiens (Human)) | BDBM50095287 (CHEMBL3085880) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Ljubljana Curated by ChEMBL | Assay Description Modulation of human Nav1.7 by automated patch clamp electrophysiology assay | Eur J Med Chem 70: 154-64 (2013) Article DOI: 10.1016/j.ejmech.2013.07.034 BindingDB Entry DOI: 10.7270/Q2DR2ZF3 | |||||||||||
More data for this Ligand-Target Pair |