BindingDB PrimarySearch

Found 2 hits Enz. Inhib. hit(s) with Target = 'Solute carrier family 22 member 3' and Ligand = 'BDBM50149890'
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Solute carrier family 22 member 3 (Homo sapiens (Human))	BDBM50149890 (CHEMBL9324 \| tetraethylammonium) Show SMILES CC[N+](CC)(CC)CC Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL DrugBank KEGG MMDB PC cid PC sid UniChem Patents Similars	Article PubMed	1.37E+6	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Medical College of Georgia Curated by ChEMBL					Assay Description TP_TRANSPORTER: inhibition of MPP+ uptake in OCT3-expressing HRPE cells				Am J Physiol Renal Physiol 279: 449-58 (2000) Article DOI: 10.1152/ajprenal.2000.279.3.f449 BindingDB Entry DOI: 10.7270/Q2708482
Medical College of Georgia Curated by ChEMBL					More data for this Ligand-Target Pair
Solute carrier family 22 member 3 (Homo sapiens (Human))	BDBM50149890 (CHEMBL9324 \| tetraethylammonium) Show SMILES CC[N+](CC)(CC)CC Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL DrugBank KEGG MMDB PC cid PC sid UniChem Patents Similars	PubMed	n/a	n/a	1.03E+7	n/a	n/a	n/a	n/a	n/a	n/a
Universidade do Porto Curated by ChEMBL					Assay Description TP_TRANSPORTER: inhibition of MPP+ uptake (MPP+: 0.2 uM) in OCT3-expressing HEK293 cells				Naunyn Schmiedebergs Arch Pharmacol 363: 40-9 (2001) BindingDB Entry DOI: 10.7270/Q2GQ702R
Universidade do Porto Curated by ChEMBL					More data for this Ligand-Target Pair