Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Somatostatin receptor type 3 (Homo sapiens (Human)) | BDBM50326873 (3-amino-N-((2S,3R,4S,5S,6R)-6-((4-chlorobenzyloxy)...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 6.33E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Alchemia Ltd Curated by ChEMBL | Assay Description Displacement of [125I]iodotyrosyl from human SST3 receptor expressed in CHO cells | J Med Chem 53: 5576-86 (2010) Article DOI: 10.1021/jm1002777 BindingDB Entry DOI: 10.7270/Q2QC03QK | |||||||||||
More data for this Ligand-Target Pair |