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Compile Data Set for Download or QSAR

Found 2 hits Enz. Inhib. hit(s) with Target = 'Somatostatin receptor type 4' and Ligand = 'BDBM506589'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Somatostatin receptor type 4


(Homo sapiens (Human))
BDBM506589
PNG
(US11045457, Example 190)
Show SMILES C[C@H]1CNCC[C@@H]1NC(=O)C(C)(C)COc1ccccc1Cl |r|
PDB

KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
n/an/a 25.1n/an/an/an/an/an/a


TBA

Assay Description
This membrane-based assay measures the ability of compounds to competitively inhibit binding of I-125 labeled somatostatin to SSTR4 in membranes from...


Citation and Details

BindingDB Entry DOI: 10.7270/Q2CN7721
More data for this
Ligand-Target Pair
Somatostatin receptor type 4


(Homo sapiens (Human))
BDBM506589
PNG
(US11045457, Example 190)
Show SMILES C[C@H]1CNCC[C@@H]1NC(=O)C(C)(C)COc1ccccc1Cl |r|
PDB

KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
n/an/an/an/a 0.158n/an/an/an/a


TBA

Assay Description
This cell-based assay measures the ability of compounds to inhibit forskolin stimulated cAMP in CHO-K1 cells overexpressing SSTR4. CHO-K1 cells overe...


Citation and Details

BindingDB Entry DOI: 10.7270/Q2CN7721
More data for this
Ligand-Target Pair