Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Substance-K receptor (HAMSTER) | BDBM50001451 (3-Amino-N-(1-{1-[1-({[1-(1-carbamoyl-3-methylsulfa...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 6 | n/a | n/a | n/a | n/a | n/a | n/a |
Marion Merrell Dow Research Institute Curated by ChEMBL | Assay Description Competitive inhibition of [125I]NKA binding to hamster urinary bladder Tachykinin receptor 2 | J Med Chem 35: 3949-55 (1992) BindingDB Entry DOI: 10.7270/Q2FF3SZB | |||||||||||
More data for this Ligand-Target Pair |