Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Substance-P receptor (Rattus norvegicus (rat)) | BDBM50229589 (Arg-Pro-Lys-Pro-Ala-Gln-Phe-Phe-Gly-Leu-Met-NH2 | ...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.740 | n/a | n/a | n/a | n/a | n/a | n/a |
Mississippi State University Curated by ChEMBL | Assay Description Displacement of [125I]Lys3-substance P from rat NK1 receptor expressed in CHO cells | J Med Chem 50: 6501-6 (2007) Article DOI: 10.1021/jm070577s BindingDB Entry DOI: 10.7270/Q2RX9BT2 | |||||||||||
More data for this Ligand-Target Pair |