Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Succinate receptor 1' and Ligand = 'BDBM50393140'   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Succinate receptor 1 (Homo sapiens (Human))	BDBM50393140 (CHEMBL2153472) Show SMILES Fc1ccc(cc1C(F)(F)F)-n1cc(CNC(=O)CCCc2ccc3cccnc3n2)cn1 Show InChI InChI=1S/C23H19F4N5O/c24-20-9-8-18(11-19(20)23(25,26)27)32-14-15(13-30-32)12-29-21(33)5-1-4-17-7-6-16-3-2-10-28-22(16)31-17/h2-3,6-11,13-14H,1,4-5,12H2,(H,29,33)	Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	210	n/a	n/a	n/a	n/a	n/a	n/a
Advinus Therapeutics Curated by ChEMBL					Assay Description Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...				Bioorg Med Chem Lett 21: 3596-602 (2011) Article DOI: 10.1016/j.bmcl.2011.04.091 BindingDB Entry DOI: 10.7270/Q2BK1DG6
					More data for this Ligand-Target Pair