Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Thrombopoietin receptor (Homo sapiens (Human)) | BDBM50219633 (4-(6-(azetidin-1-yl)pyrimidin-4-ylamino)-N-(4-(2-f...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 23 | n/a | n/a | n/a | n/a |
Pfizer Global Research & Development Curated by ChEMBL | Assay Description Agonist activity at human TPOr expressed in BaF3 cells by reporter assay | Bioorg Med Chem Lett 17: 5447-54 (2007) Article DOI: 10.1016/j.bmcl.2007.07.038 BindingDB Entry DOI: 10.7270/Q2Q52PBC | |||||||||||
More data for this Ligand-Target Pair |