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Found 1 hit Enz. Inhib. hit(s) with Target = 'Thromboxane A2 receptor' and Ligand = 'BDBM50002819'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Thromboxane A2 receptor


(Homo sapiens (Human))		BDBM50002819
PNG
(11-(2-Naphtho[2,3-d]imidazol-1-yl-ethylidene)-6,11...)
Show SMILES OC(=O)c1ccc2OCc3ccccc3\C(=C/Cn3cnc4cc5ccccc5cc34)c2c1
Show InChI InChI=1S/C28H20N2O3/c31-28(32)20-9-10-27-24(13-20)23(22-8-4-3-7-21(22)16-33-27)11-12-30-17-29-25-14-18-5-1-2-6-19(18)15-26(25)30/h1-11,13-15,17H,12,16H2,(H,31,32)/b23-11+
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PC sid
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Similars
PubMed
 280n/an/an/an/an/an/an/an/a



Kyowa Hakko Kogyo Company, Ltd.

Curated by ChEMBL


Assay Description
Binding affinity at TXA2/PGH2 receptor by measuring its ability to displace [3H]-U-46,619 from guinea pig platelets

J Med Chem 35: 3402-13 (1992)


BindingDB Entry DOI: 10.7270/Q2J38RG1
More data for this
Ligand-Target Pair