Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Trace amine-associated receptor 1 (Rattus norvegicus (Rat)) | BDBM167503 (US9073911, 52) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 7.40 | n/a | n/a | n/a | n/a | n/a | n/a | 7.4 | n/a |
HOFFMANN-LA ROCHE INC. US Patent | Assay Description The TAAR1 radioligand 3[H](S)-4-[(ethyl-phenyl-amino)-methyl]-4,5-dihydro-oxazol-2-ylamine (described in WO 2008/098857) was used at a concentration ... | US Patent US9073911 (2015) BindingDB Entry DOI: 10.7270/Q2N29VPX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Trace amine-associated receptor 1 (Mus musculus (Mouse)) | BDBM167503 (US9073911, 52) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 8.40 | n/a | n/a | n/a | n/a | n/a | n/a | 7.4 | n/a |
HOFFMANN-LA ROCHE INC. US Patent | Assay Description The TAAR1 radioligand 3[H](S)-4-[(ethyl-phenyl-amino)-methyl]-4,5-dihydro-oxazol-2-ylamine (described in WO 2008/098857) was used at a concentration ... | US Patent US9073911 (2015) BindingDB Entry DOI: 10.7270/Q2N29VPX | |||||||||||
More data for this Ligand-Target Pair |