Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Transcription activator BRG1 [1448-1575]' and Ligand = 'BDBM394510'   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Transcription activator BRG1 [1448-1575] (Homo sapiens (Human))	BDBM394510 (2-(6-amino-5-(4- | US10308614, Example 111) Show SMILES CC1CN(CCN1S(=O)(=O)C1CC1)c1cc(nnc1N)-c1ccccc1O Show InChI InChI=1S/C18H23N5O3S/c1-12-11-22(8-9-23(12)27(25,26)13-6-7-13)16-10-15(20-21-18(16)19)14-4-2-3-5-17(14)24/h2-5,10,12-13,24H,6-9,11H2,1H3,(H2,19,21)	PDB MMDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	19.7	n/a	n/a	n/a	n/a	n/a	n/a
The Institute of Cancer Research					Assay Description His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvpr\gsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNA...				J Med Chem 52: 2255-64 (2009) BindingDB Entry DOI: 10.7270/Q26112NJ
					More data for this Ligand-Target Pair