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Found 1 hit Enz. Inhib. hit(s) with Target = 'Transcription activator BRG1 [1448-1575]' and Ligand = 'BDBM394575'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Transcription activator BRG1 [1448-1575]


(Homo sapiens (Human))		BDBM394575
PNG
(2-(6-amino-5-(2- | US10308614, Example 178)
Show SMILES CC(COc1cc(nnc1N)-c1ccccc1O)c1ccccc1
Show InChI InChI=1S/C19H19N3O2/c1-13(14-7-3-2-4-8-14)12-24-18-11-16(21-22-19(18)20)15-9-5-6-10-17(15)23/h2-11,13,23H,12H2,1H3,(H2,20,22)
PDB
MMDB

KEGG

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
n/an/a 12.2n/an/an/an/an/an/a



The Institute of Cancer Research



Assay Description
His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvpr\gsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNA...

J Med Chem 52: 2255-64 (2009)


BindingDB Entry DOI: 10.7270/Q26112NJ
More data for this
Ligand-Target Pair