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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Transcription factor 4' and Ligand = 'BDBM50500848'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Transcription factor 4


(Homo sapiens)		BDBM50500848
PNG
(CHEMBL2397075)
Show SMILES COc1cc(O)c2c3c1c1c(OC)cc(O)c4c1c(c(CC(C)OC(=O)c1c(C)cc(O)cc1O)c(OC)c4=O)c3c(CC(C)OC(=O)c1c(C)cc(O)cc1O)c(OC)c2=O
Show InChI InChI=1S/C46H42O16/c1-17-9-21(47)13-25(49)31(17)45(55)61-19(3)11-23-33-34-24(12-20(4)62-46(56)32-18(2)10-22(48)14-26(32)50)44(60-8)42(54)36-28(52)16-30(58-6)38(40(34)36)37-29(57-5)15-27(51)35(39(33)37)41(53)43(23)59-7/h9-10,13-16,19-20,47-52H,11-12H2,1-8H3
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 4.10E+3n/an/an/an/an/an/a



King Saud University

Curated by ChEMBL


Assay Description
Inhibition of human GST tagged Tcf4/beta catenin interaction after 2 hrs using fluorescent AP Attophos substrate by ELISA analysis

Bioorg Med Chem Lett 26: 1664-70 (2016)


Article DOI: 10.1016/j.bmcl.2016.02.064
BindingDB Entry DOI: 10.7270/Q25H7K8M
More data for this
Ligand-Target Pair