Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Transient receptor potential cation channel subfamily M member 4' and Ligand = 'BDBM50526040'   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Transient receptor potential cation channel subfamily M member 4 (Homo sapiens)	BDBM50526040 (CHEMBL4447880) Show SMILES Clc1ccc(C(=O)NS(=O)(=O)C2CC2)c(NC(=O)COc2ccccc2Cl)c1 Show InChI InChI=1S/C18H16Cl2N2O5S/c19-11-5-8-13(18(24)22-28(25,26)12-6-7-12)15(9-11)21-17(23)10-27-16-4-2-1-3-14(16)20/h1-5,8-9,12H,6-7,10H2,(H,21,23)(H,22,24)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	2.80E+3	n/a	n/a	n/a	n/a	n/a	n/a
University of Berne Curated by ChEMBL					Assay Description Inhibition of Flag-tagged TRPM4 (unknown origin) expressed in HEK293 cells assessed as reduction in intracellular Na+ influx after 45 mins by ANG2 dy...				Eur J Med Chem 166: 167-177 (2019) Article DOI: 10.1016/j.ejmech.2019.01.048 BindingDB Entry DOI: 10.7270/Q2GH9NCB
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