Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Transient receptor potential cation channel subfamily M member 8' and Ligand = 'BDBM50268809'   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Transient receptor potential cation channel subfamily M member 8 (Homo sapiens (Human))	BDBM50268809 (CHEMBL4094279) Show SMILES Cc1ccc(OCC(=O)N(O)Cc2cccs2)cc1 Show InChI InChI=1S/C14H15NO3S/c1-11-4-6-12(7-5-11)18-10-14(16)15(17)9-13-3-2-8-19-13/h2-8,17H,9-10H2,1H3	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	8.00E+3	n/a	n/a	n/a	n/a
Senomyx Inc., 4767 Nexus Centre Dr, San Diego, CA 92121, United States. Curated by ChEMBL					Assay Description Agonist activity at human TRPM8 expressed in HEK293 cells assessed as increase in intracellular calcium level after 15 mins by Fluo-3-AM dye-based fl...				Bioorg Med Chem Lett 27: 3931-3938 (2017) Article DOI: 10.1016/j.bmcl.2017.04.003 BindingDB Entry DOI: 10.7270/Q25H7JRG
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