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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Transient receptor potential cation channel subfamily M member 8' and Ligand = 'BDBM50269670'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Transient receptor potential cation channel subfamily M member 8


(Homo sapiens (Human))		BDBM50269670
PNG
(CHEMBL4072058)
Show SMILES CCCCOCCOC(C(C)Oc1c(OC)cc(CC=C)cc1OC)c1ccc(O)c(OC)c1
Show InChI InChI=1S/C27H38O7/c1-7-9-13-32-14-15-33-26(21-11-12-22(28)23(18-21)29-4)19(3)34-27-24(30-5)16-20(10-8-2)17-25(27)31-6/h8,11-12,16-19,26,28H,2,7,9-10,13-15H2,1,3-6H3
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PC cid
PC sid
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Similars
Article
PubMed
n/an/an/an/a 153n/an/an/an/a



Kansei Science Research and Biological Science Research, Kao Corporation, 2606 Akabane, Ichikai-Machi, Haga-Gun, Tochigi 321-3497, Japan.

Curated by ChEMBL


Assay Description
Agonist activity at full length recombinant human TRPM8 expressed in HEK293 cells assessed as increase in intracellular Ca2+ level pre-incubated for ...

ACS Med Chem Lett 8: 715-719 (2017)


Article DOI: 10.1021/acsmedchemlett.7b00104
BindingDB Entry DOI: 10.7270/Q2CZ39N2
More data for this
Ligand-Target Pair