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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Transient receptor potential cation channel subfamily V member 1/2/4' and Ligand = 'BDBM50222692'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Transient receptor potential cation channel subfamily V member 1/2/4


(Rattus norvegicus-Rattus norvegicus (rat))		BDBM50222692
PNG
(CHEMBL348634)
Show SMILES CCCCCCCCN(CCCc1ccc(O)c(OC)c1)C(\S)=N\CCc1ccccc1
Show InChI InChI=1S/C27H40N2O2S/c1-3-4-5-6-7-11-20-29(27(32)28-19-18-23-13-9-8-10-14-23)21-12-15-24-16-17-25(30)26(22-24)31-2/h8-10,13-14,16-17,22,30H,3-7,11-12,15,18-21H2,1-2H3,(H,28,32)
PDB

UniProtKB/SwissProt

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PC cid
PC sid
UniChem

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Similars
PubMed
n/an/a>30n/an/an/an/an/an/a



Seoul National University

Curated by ChEMBL


Assay Description
Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...

Bioorg Med Chem Lett 13: 601-4 (2003)


BindingDB Entry DOI: 10.7270/Q2XP7747
More data for this
Ligand-Target Pair