Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Transient receptor potential cation channel subfamily V member 1' and Ligand = 'BDBM128053'   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Transient receptor potential cation channel subfamily V member 1 (Homo sapiens (Human))	BDBM128053 (US8796328, 31) Show SMILES CS(=O)(=O)Nc1ccc(CNC(=O)N[C@@H]2CCOc3c2cccc3C(F)(F)F)cc1F Show InChI InChI=1S/C19H19F4N3O4S/c1-31(28,29)26-16-6-5-11(9-14(16)20)10-24-18(27)25-15-7-8-30-17-12(15)3-2-4-13(17)19(21,22)23/h2-6,9,15,26H,7-8,10H2,1H3,(H2,24,25,27)/t15-/m1/s1	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	3.80E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA US Patent					Assay Description The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...				US Patent US8796328 (2014) BindingDB Entry DOI: 10.7270/Q2639NFM
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