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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Type-1 angiotensin II receptor' and Ligand = 'BDBM50282438'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Type-1 angiotensin II receptor


(RABBIT)		BDBM50282438
PNG
(CHEMBL352137 | Quinazolinone Biphenyl Acylsulfonam...)
Show SMILES CCCCc1nc2ccc(cc2c(=O)n1Cc1ccc(cc1)-c1ccccc1S(=O)(=O)NC(=O)NC(C)C)C(C)C
Show InChI InChI=1S/C32H38N4O4S/c1-6-7-12-30-34-28-18-17-25(21(2)3)19-27(28)31(37)36(30)20-23-13-15-24(16-14-23)26-10-8-9-11-29(26)41(39,40)35-32(38)33-22(4)5/h8-11,13-19,21-22H,6-7,12,20H2,1-5H3,(H2,33,35,38)
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PC cid
PC sid
UniChem

Similars
Article
n/an/a 5.60n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
In vitro displacement of 125I-[Sar1, Ile8] from AT1 receptors in rabbit aorta membrane

Bioorg Med Chem Lett 4: 75-80 (1994)


Article DOI: 10.1016/S0960-894X(01)81125-2
BindingDB Entry DOI: 10.7270/Q2J1033H
More data for this
Ligand-Target Pair