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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Type-1 angiotensin II receptor' and Ligand = 'BDBM50284464'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Type-1 angiotensin II receptor


(RABBIT)		BDBM50284464
PNG
(CHEMBL15788 | [4-(2-Ethyl-5,7-dimethyl-imidazo[4,5...)
Show SMILES CCCc1cc(Cn2c(CC)nc3c(C)cc(C)nc23)ccc1OC(C(O)=O)c1ccccc1C
Show InChI InChI=1S/C29H33N3O3/c1-6-10-22-16-21(17-32-25(7-2)31-26-19(4)15-20(5)30-28(26)32)13-14-24(22)35-27(29(33)34)23-12-9-8-11-18(23)3/h8-9,11-16,27H,6-7,10,17H2,1-5H3,(H,33,34)
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Article
n/an/a 11n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Tested for its ability to displace the specific binding ligand [125I]-Sar 1,lle8-AlI from rabbit aortic membrane (AT1 receptor)

Bioorg Med Chem Lett 5: 1151-1154 (1995)


Article DOI: 10.1016/0960-894X(95)00185-V
BindingDB Entry DOI: 10.7270/Q2J67GV9
More data for this
Ligand-Target Pair