Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Tyrosine-protein kinase Lck (Homo sapiens (Human)) | BDBM50037419 (5-Methoxy-8-nitro-2-(4-nitro-phenyl)-chromen-4-one...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | >2.00E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
Purdue University Curated by ChEMBL | Assay Description In vitro inhibition of protein-tyrosine activity of p56lck enzyme in presence of 50 uM ATP | J Med Chem 37: 3353-62 (1994) BindingDB Entry DOI: 10.7270/Q2D21WNP | |||||||||||
More data for this Ligand-Target Pair |