Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Tyrosine-protein kinase Lck (Homo sapiens (Human)) | BDBM50413752 (CHEMBL2012519 | L-783277) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 750 | n/a | n/a | n/a | n/a | n/a | n/a |
AMRI Curated by ChEMBL | Assay Description Inhibition of LCK (unknown origin) | Bioorg Med Chem Lett 19: 3059-62 (2009) Article DOI: 10.1016/j.bmcl.2009.04.005 BindingDB Entry DOI: 10.7270/Q2MG7PDB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tyrosine-protein kinase Lck (Homo sapiens (Human)) | BDBM50413752 (CHEMBL2012519 | L-783277) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of LCK by TR-FRET based LanthaScreen assay | ACS Med Chem Lett 2: 22-27 (2011) Article DOI: 10.1021/ml1001807 BindingDB Entry DOI: 10.7270/Q2542NWT | |||||||||||
More data for this Ligand-Target Pair |