Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Tyrosine-protein kinase receptor TYRO3 (Homo sapiens (Human)) | BDBM50059889 ((staurosporine)3-methoxy-2-methyl-4-methylamino-(2...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 49.0 | n/a | n/a | n/a | n/a | n/a | n/a |
Centre Universitaire Curated by ChEMBL | Assay Description Inhibition of TYRO3/SKY | Eur J Med Chem 45: 3389-93 (2010) Article DOI: 10.1016/j.ejmech.2010.04.026 BindingDB Entry DOI: 10.7270/Q2TH8MWC | |||||||||||
More data for this Ligand-Target Pair |