Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
UDP-glucuronosyltransferase 1A1 (Homo sapiens (Human)) | BDBM50460861 (CHEMBL4229237) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >2.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck & Co. Curated by ChEMBL | Assay Description Inhibition of UGT1A1 in human liver microsomes assessed as decrease in estradiol-3 glucuronidation | Bioorg Med Chem Lett 28: 1392-1396 (2018) Article DOI: 10.1016/j.bmcl.2018.02.039 BindingDB Entry DOI: 10.7270/Q25T3P36 | |||||||||||
More data for this Ligand-Target Pair |