Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Vascular endothelial growth factor receptor 2 (Homo sapiens (Human)) | BDBM50192487 ((7,8-dimethoxy-10,11-dihydro-5H-2,4,5,11-tetraaza-...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
ImClone Systems Inc Curated by ChEMBL | Assay Description Inhibition of KDR measured as pGAT-biotin peptide phosphorylation by HTRF assay | Bioorg Med Chem Lett 16: 5102-6 (2006) Article DOI: 10.1016/j.bmcl.2006.07.031 BindingDB Entry DOI: 10.7270/Q2K9374T | |||||||||||
More data for this Ligand-Target Pair |