Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Vascular endothelial growth factor receptor 2 (Homo sapiens (Human)) | BDBM50318959 (CHEMBL1084337 | rac-9-isobutyl-5-methyl-12-(tetrah...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | n/a |
Cephalon, Inc. Curated by ChEMBL | Assay Description Inhibition of VEGF-stimulated VEGFR2 autophosphorylation in HUVEC | Bioorg Med Chem Lett 20: 3356-60 (2010) Article DOI: 10.1016/j.bmcl.2010.04.021 BindingDB Entry DOI: 10.7270/Q2HT2PH9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vascular endothelial growth factor receptor 2 (Homo sapiens (Human)) | BDBM50318959 (CHEMBL1084337 | rac-9-isobutyl-5-methyl-12-(tetrah...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 11 | n/a | n/a | n/a | n/a | n/a | n/a |
Cephalon, Inc. Curated by ChEMBL | Assay Description Inhibition of human recombinant VEGFR2 by time resolved fluorescence measurements | Bioorg Med Chem Lett 20: 3356-60 (2010) Article DOI: 10.1016/j.bmcl.2010.04.021 BindingDB Entry DOI: 10.7270/Q2HT2PH9 | |||||||||||
More data for this Ligand-Target Pair |