Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Vasopressin V1a/V1b receptor (Homo sapiens (Human)) | BDBM50137948 (Biphenyl-2-carboxylic acid [2-[3-(4-methyl-[1,4]di...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | <1 | n/a | n/a | n/a | n/a | n/a | n/a |
Central Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in human platelet | J Med Chem 47: 101-9 (2003) Article DOI: 10.1021/jm030287l BindingDB Entry DOI: 10.7270/Q2TX3DT7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vasopressin V1a/V1b receptor (RAT) | BDBM50137948 (Biphenyl-2-carboxylic acid [2-[3-(4-methyl-[1,4]di...) | MMDB UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
Central Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liver | J Med Chem 47: 101-9 (2003) Article DOI: 10.1021/jm030287l BindingDB Entry DOI: 10.7270/Q2TX3DT7 | |||||||||||
More data for this Ligand-Target Pair |