BindingDB PrimarySearch

Found 2 hits Enz. Inhib. hit(s) with Target = 'Voltage-dependent T-type calcium channel subunit alpha-1G' and Ligand = 'BDBM50148177'
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Voltage-dependent T-type calcium channel subunit alpha-1G (Homo sapiens (Human))	BDBM50148177 (CHEMBL115159 \| KYS-05040 \| N-(4-Amino-benzyl)-2-(3...) Show SMILES Show InChI	PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	1.30E+4	n/a	n/a	n/a	n/a	n/a	n/a
Kyung Hee University Curated by ChEMBL					Assay Description Inhibition of human T-type calcium channel alpha1G in HEK293 cells				Bioorg Med Chem Lett 20: 38-41 (2010) Article DOI: 10.1016/j.bmcl.2009.11.049 BindingDB Entry DOI: 10.7270/Q2MS3V0M
Kyung Hee University Curated by ChEMBL					More data for this Ligand-Target Pair
Voltage-dependent T-type calcium channel subunit alpha-1G (Homo sapiens (Human))	BDBM50148177 (CHEMBL115159 \| KYS-05040 \| N-(4-Amino-benzyl)-2-(3...) Show SMILES Show InChI	PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	1.44E+4	n/a	n/a	n/a	n/a	n/a	n/a
Institute of Science & Technology Curated by ChEMBL					Assay Description Concentration of the compounds required for inhibition of HEK293 cells (alpha1G T-type)				Bioorg Med Chem Lett 14: 3379-84 (2004) Article DOI: 10.1016/j.bmcl.2004.04.090 BindingDB Entry DOI: 10.7270/Q21Z43VJ
Institute of Science & Technology Curated by ChEMBL					More data for this Ligand-Target Pair