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Found 1 hit Enz. Inhib. hit(s) with Target = 'Voltage-dependent T-type calcium channel subunit alpha-1H' and Ligand = 'BDBM372619'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Voltage-dependent T-type calcium channel subunit alpha-1H


(Homo sapiens (Human))		BDBM372619
PNG
(N-[2-(4-Difluoromethoxy-3-fluoro-benzyl)-2H-[1,2,3...)
Show SMILES Cn1ncc2cc(CC(=O)Nc3cnn(Cc4ccc(OC(F)F)c(F)c4)n3)ccc12
Show InChI InChI=1S/C20H17F3N6O2/c1-28-16-4-2-12(6-14(16)9-24-28)8-19(30)26-18-10-25-29(27-18)11-13-3-5-17(15(21)7-13)31-20(22)23/h2-7,9-10,20H,8,11H2,1H3,(H,26,27,30)
PDB

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PC cid
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US Patent
n/an/a 22n/an/an/an/an/an/a



University of Alberta



Assay Description
Stock solutions of test compounds are prepared to a concentration of 10 mM in DMSO. For the Cav3.2 assay, serial dilutions of the compounds are prepa...

J Med Chem 49: 1668-83 (2006)


BindingDB Entry DOI: 10.7270/Q2794709
More data for this
Ligand-Target Pair