Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Voltage-dependent T-type calcium channel subunit alpha-1H (Homo sapiens (Human)) | BDBM50095309 (CHEMBL3589557) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
AbbVie, Inc. Curated by ChEMBL | Assay Description Inhibition of human recombinant Cav3.2 channel | ACS Med Chem Lett 6: 641-4 (2015) Article DOI: 10.1021/acsmedchemlett.5b00023 BindingDB Entry DOI: 10.7270/Q27D2WW3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Voltage-dependent T-type calcium channel subunit alpha-1H (Rattus norvegicus) | BDBM50095309 (CHEMBL3589557) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 7.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
AbbVie, Inc. Curated by ChEMBL | Assay Description Inhibition of Cav3.2 channel in rat DRG neurons assessed as reduction in LVA currents | ACS Med Chem Lett 6: 641-4 (2015) Article DOI: 10.1021/acsmedchemlett.5b00023 BindingDB Entry DOI: 10.7270/Q27D2WW3 | |||||||||||
More data for this Ligand-Target Pair |