BindingDB logo
myBDB logout
Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'cAMP-specific 3',5'-cyclic phosphodiesterase 4B' and Ligand = 'BDBM50558597'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
cAMP-specific 3',5'-cyclic phosphodiesterase 4B


(Homo sapiens (Human))
BDBM50558597
PNG
(CHEMBL4787884)
Show SMILES FC(F)Oc1ccc(-c2nc(cs2)C(=O)Nc2c(Cl)cncc2Cl)c2c3ccccc3oc12
PDB

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 127n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of human PDE4B using [3H]cAMP as substrate incubated for 5 mins followed by substrate addition and measured after 10 mins by scintillation...


Citation and Details

Article DOI: 10.1016/j.bmc.2016.09.011
BindingDB Entry DOI: 10.7270/Q2N58R28
More data for this
Ligand-Target Pair