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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'cGMP-dependent protein kinase' and Ligand = 'BDBM340882'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
cGMP-dependent protein kinase


()		BDBM340882
PNG
(3-isopropyl-1-(quinolin-3-yl)imidazo[1,5- a]pyrazi...)
Show SMILES CC(C)c1nc(-c2cnc3ccccc3c2)c2c(N)nccn12
Show InChI InChI=1S/C18H17N5/c1-11(2)18-22-15(16-17(19)20-7-8-23(16)18)13-9-12-5-3-4-6-14(12)21-10-13/h3-11H,1-2H3,(H2,19,20)
UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
n/an/a 40n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of TgCDPK1 and CpCDPK1 was determined using a luminescent kinase assay which measures ATP depletion in the presence of the Syntide 2 pepti...

Citation and Details

BindingDB Entry DOI: 10.7270/Q2K077GQ
More data for this
Ligand-Target Pair