Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
cGMP-dependent protein kinase () | BDBM50345749 (3-(3-(benzyloxy)phenyl)-1-isopropyl-1H-pyrazolo[3,...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 1.06E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of TgCDPK1 and CpCDPK1 was determined using a luminescent kinase assay which measures ATP depletion in the presence of the Syntide 2 pepti... | Citation and Details BindingDB Entry DOI: 10.7270/Q2K077GQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cGMP-dependent protein kinase () | BDBM50345749 (3-(3-(benzyloxy)phenyl)-1-isopropyl-1H-pyrazolo[3,...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 1.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Kinase phosphorylation reactions were performed in a buffered medium containing 20 mM HEPES pH 7.5 (KOH), 0.1% BSA, 10 mM MgCl2, 1 mM EGTA (pH 7.2), ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2K077GQ | |||||||||||
More data for this Ligand-Target Pair |