Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
cGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B (Homo sapiens (Human)) | BDBM50287548 (5-Phenyl-3-propyl-1,6-dihydro-pyrazolo[4,3-d]pyrim...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 6.30E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of Phosphodiesterase 3 from rabbit platelets | Bioorg Med Chem Lett 6: 1819-1824 (1996) Article DOI: 10.1016/0960-894X(96)00323-X BindingDB Entry DOI: 10.7270/Q2G73DQW | |||||||||||
More data for this Ligand-Target Pair |