Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sodium channel protein type 1/2/3 subunit alpha (Rattus norvegicus) | BDBM50003560 (4-methoxy-17-methyl-17-azatetracyclo[7.5.3.01,10.0...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 1.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Pharmacia& Upjohn Curated by ChEMBL | Assay Description Binding of [3H]batrachotoxin (BTX) to rat brain sodium channel | Bioorg Med Chem Lett 9: 1783-8 (1999) BindingDB Entry DOI: 10.7270/Q28K7C8R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1 (Mus musculus (Mouse)-MOUSE) | BDBM50003560 (4-methoxy-17-methyl-17-azatetracyclo[7.5.3.01,10.0...) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 2.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Concentration required to inhibit [3H]naltrexone binding to Opioid receptors | J Med Chem 25: 1264-6 (1982) BindingDB Entry DOI: 10.7270/Q29P33VW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium channel protein type 1/2/3 subunit alpha (Rattus norvegicus) | BDBM50003560 (4-methoxy-17-methyl-17-azatetracyclo[7.5.3.01,10.0...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | >3.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Pharmacia& Upjohn Curated by ChEMBL | Assay Description Binding of [3H]saxitoxin (STX) to rat brain sodium channel | Bioorg Med Chem Lett 9: 1783-8 (1999) BindingDB Entry DOI: 10.7270/Q28K7C8R | |||||||||||
More data for this Ligand-Target Pair |