BindingDB PrimarySearch

Found 4 hits of ic50 for UniProtKB: P09482
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Neuronal acetylcholine receptor subunit alpha-4 (Gallus gallus)	BDBM50251867 (CHEMBL518310 \| N-(3-((6-chloropyridin-3-yl)methyl)...) Show SMILES FC(F)(F)C(=O)\N=c1/sccn1Cc1ccc(Cl)nc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	500	n/a	n/a	n/a	n/a	n/a	n/a
University of California Curated by ChEMBL					Assay Description Displacement of [3H]nicotine from chick alpha4beta2 nAChR				J Med Chem 51: 4213-8 (2008) Article DOI: 10.1021/jm800191a BindingDB Entry DOI: 10.7270/Q2D21XDZ
University of California Curated by ChEMBL					More data for this Ligand-Target Pair
Neuronal acetylcholine receptor subunit alpha-4 (Gallus gallus)	BDBM50251868 ((Z)-thiacloprid \| CHEMBL451432 \| {(2Z)-3-[(6-chlor...) Show SMILES Clc1ccc(CN2CCS\C2=N/C#N)cn1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid PDB UniChem Patents Similars	Article PubMed	n/a	n/a	860	n/a	n/a	n/a	n/a	n/a	n/a
University of California Curated by ChEMBL					Assay Description Displacement of [3H]nicotine from chick alpha4beta2 nAChR				J Med Chem 51: 4213-8 (2008) Article DOI: 10.1021/jm800191a BindingDB Entry DOI: 10.7270/Q2D21XDZ
University of California Curated by ChEMBL					More data for this Ligand-Target Pair
Neuronal acetylcholine receptor subunit alpha-4 (Gallus gallus)	BDBM50252631 (CHEMBL494278 \| N-(3-((6-chloropyridin-3-yl)methyl)...) Show SMILES Clc1ccc(Cn2ccs\c2=N/C(=O)c2cnccn2)cn1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	900	n/a	n/a	n/a	n/a	n/a	n/a
University of California Curated by ChEMBL					Assay Description Displacement of [3H]nicotine from chick alpha4beta2 nAChR				J Med Chem 51: 4213-8 (2008) Article DOI: 10.1021/jm800191a BindingDB Entry DOI: 10.7270/Q2D21XDZ
University of California Curated by ChEMBL					More data for this Ligand-Target Pair
Neuronal acetylcholine receptor subunit alpha-4 (Gallus gallus)	BDBM50212288 ((2E)-1-[(6-chloropyridin-3-yl)methyl]-N-nitroimida...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid PDB UniChem Patents Similars	Article PubMed	n/a	n/a	2.60E+3	n/a	n/a	n/a	n/a	n/a	n/a
University of California Curated by ChEMBL					Assay Description Displacement of [3H]nicotine from chick alpha4beta2 nAChR				J Med Chem 51: 4213-8 (2008) Article DOI: 10.1021/jm800191a BindingDB Entry DOI: 10.7270/Q2D21XDZ
University of California Curated by ChEMBL					More data for this Ligand-Target Pair